Kuiyong Dong^†, Bin Yan^‡, Sailan Chang^†, Yongjian Chi^†, Lihua Qiu^*†（邱丽华）, and Xinfang Xu^*†（徐新芳）

^† Key Laboratory of Organic Synthesis of Jiangsu Province, College of Chemistry, Chemical Engineering and Materials Science, Soochow University, Suzhou 215123, China

^‡ Jinghua Anti-cancer Pharmaceutical Engineering Center, Nantong 226407, China

J. Org. Chem., 2016, 81 (15), pp 6887–6892

An efficient transition-metal-free fluoroarylation reaction of N-aryl diazoacetamides with NFSI (N-fluorobenzenesulfonimide) is described. This reaction directly provides 3-fluorooxindole derivatives in yields of 67–93% with high selectivity via a carbene-free process under mild reaction conditions.

链接：http://pubs.acs.org/doi/abs/10.1021/acs.joc.6b01286