Cu(acac)2∙H2O-Catalyzed Sonogashira-Type Couplings of Aryl Halides and Terminal Alkynes
Cu(acac)2∙H2O-Catalyzed Sonogashira-Type Couplings of Aryl Halides and Terminal Alkynes
Tingyi Li, Xiaoming Qu, Guanlei Xie, Prof. Jincheng Mao*
DOI: 10.1002/asia.201000923


Graphical Abstract

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Highly selective coupling of aryl halides with terminal alkynes can be conducted using low-cost and readily available [Cu(acac)2]H2O under palladium- and amine-free conditions. This protocol makes the typical Sonogashira reaction more practical and useful (TBAB=tetrabutyl ammonium bromide; DMSO=dimethyl sulfoxide; see scheme).